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1

2,3-Diaminopyridine as a platform for designing structurally unique nonpeptide bradykinin B1 receptor antagonists

Dong-Mei Feng, Jenny M. Wai, Scott D. Kuduk, Christina Ng, Kathy L. Murphy, Richard W. Ransom, Duane Reiss, Raymond S.L. Chang, Charles M. Harrell, Tanya MacNeil, Cuyue Tang, Thomayant Prueksaritanont

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 112 KB

english, 2005

2

Bradykinin B1 antagonists: Biphenyl SAR studies in the cyclopropanecarboxamide series

Scott D. Kuduk, Robert M. DiPardo, Ronald K. Chang, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone, Mark G. Bock

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2007

Langue:

english

Fichier:

PDF, 148 KB

english, 2007

3

Remarkable long range effects on the diastereoface selectivity in an aldol condensation

Christina R Harris, Scott D Kuduk, Aaron Balog, Ken A Savin, Samuel J Danishefsky

Journal:

Tetrahedron Letters

Année:

1999

Langue:

english

Fichier:

PDF, 160 KB

english, 1999

4

Tetrabutylammonium Salt Induced Denitration of Nitropyridines: Synthesis of Fluoro-, Hydroxy-, and Methoxypyridines

Kuduk, Scott D., DiPardo, Robert M., Bock, Mark G.

Journal:

Organic Letters

Année:

2005

Langue:

english

Fichier:

PDF, 61 KB

english, 2005

5

ChemInform Abstract: Synthetic and Immunological Studies on Clustered Modes of Mucin-Related Tn and TF O-Linked Antigens: The Preparation of a Glycopeptide-Based Vaccine for Clinical Trials Against Prostate Cancer.

Scott D. Kuduk, Jacob B. Schwarz, Xiao-Tao Chen, Peter W. Glunz, Dalibor Sames, Govindaswami Ragupathi, Philip O. Livingston, Samuel J. Danishefsky

Journal:

Année:

1999

Fichier:

PDF, 27 KB

1999

6

ChemInform Abstract: Remarkable Long Range Effects on the Diastereoface Selectivity in an Aldol Condensation.

Christina R. Harris, Scott D. Kuduk, Aaron Balog, Ken A. Savin, Samuel J. Danishefsky

Journal:

Année:

1999

Fichier:

PDF, 34 KB

1999

7

ChemInform Abstract: A Broadly Applicable Method for the Efficient Synthesis of α-O-Linked Glycopeptides and Clustered Sialic Acid Residues.

Jacob B. Schwarz, Scott D. Kuduk, Xiao-Tao Chen, Dalibor Sames, Peter W. Glunz, Samuel J. Danishefsky

Journal:

Année:

1999

Fichier:

PDF, 28 KB

1999

8

ChemInform Abstract: Synthesis and Evaluation of Geldanamycin-Estradiol Hybrids.

Scott D. Kuduk, Fuzhong F. Zheng, Laura Sepp-Lorenzino, Neal Rosen, Samuel J. Danishefsky

Journal:

Année:

1999

Fichier:

PDF, 30 KB

1999

9

ChemInform Abstract: Synthesis and Evaluation of Geldanamycin—Testosterone Hybrids.

Scott D. Kuduk, Christina R. Harris, Fuzhong F. Zheng, Laura Sepp-Lorenzino, Quathek Ouerfelli, Neal Rosen, Samuel J. Danishefsky

Journal:

Année:

2000

Fichier:

PDF, 25 KB

2000

10

ChemInform Abstract: Total Synthesis and Antitumor Activity of 12,13-Desoxyepothilone F: An Unexpected Solvolysis Problem at C15, Mediated by Remote Substitution at C21.

Chul Bom Lee, Ting-Chao Chou, Xiu-Guo Zhang, Zhi-Guang Wang, Scott D. Kuduk, Mark D. Chappell, Shawn J. Stachel, Samuel J. Danishefsky

Journal:

Année:

2001

Langue:

english

Fichier:

PDF, 39 KB

english, 2001

11

ChemInform Abstract: Chemical Synthesis and Biological Studies of the Epothilones: Microtubule Stabilizing Agents with Enhanced Activity Against Multidrug-Resistant Cell Lines and Tumors

Christina R. Harris, Scott D. Kuduk, Samuel J. Danishefsky

Journal:

Année:

2002

Fichier:

PDF, 25 KB

2002

12

Synthesis of 2,3-Diaminodihydropyrroles via Thioimidate Cyclopropane Rearrangement.

Scott D. Kuduk, Christina Ng, Ronald K. Chang, Mark G. Bock

Journal:

Année:

2003

Fichier:

PDF, 129 KB

2003

13

Reversal of Diastereoselection in the Addition of Grignard Reagents to Chiral 2-Pyridyl tert-Butyl (Ellman) Sulfinimines.

Scott D. Kuduk, Robert M. DiPardo, Ronald K. Chang, Christina Ng, Mark G. Bock

Journal:

Année:

2004

Fichier:

PDF, 16 KB

2004

14

Tetrabutylammonium Salt Induced Denitration of Nitropyridines: Synthesis of Fluoro-, Hydroxy-, and Methoxypyridines.

Scott D. Kuduk, Robert M. DiPardo, Mark G. Bock

Journal:

Année:

2005

Fichier:

PDF, 31 KB

2005

15

ChemInform Abstract: Preparation of 4-Heteroaryl-4-cyanopiperidines via SNAr Substitution Reactions.

Ronald K. Chang, Christina N. Di Marco, Daniel R. Pitts, Thomas J. Greshock, Scott D. Kuduk

Journal:

Année:

2010

Fichier:

PDF, 30 KB

2010

16

ChemInform Abstract: Preparation of 2,4,5-Trisubstituted Pyrazolo[4,3-c]quinolin-3-ones.

Douglas C. Beshore, Robert M. DiPardo, Scott D. Kuduk

Journal:

Année:

2010

Fichier:

PDF, 43 KB

2010

17

Syntheses of new fluorine-containing taxoids by means of β-Lactam Synthon Method

Iwao Ojima, Scott D. Kuduk, John C. Slater, Rayomand H. Gimi, Chung Ming Sun

Journal:

Année:

1996

Langue:

english

Fichier:

PDF, 1.06 MB

english, 1996

18

Pyridine containing M1 positive allosteric modulators with reduced plasma protein binding

Scott D. Kuduk, Christina N. Di Marco, Victoria Cofre, Daniel R. Pitts, William J. Ray, Lei Ma, Marion Wittmann, Matthew Seager, Kenneth Koeplinger, Chuck D. Thompson, George D. Hartman, Mark T. Bilod

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 2.57 MB

english, 2010

19

N-Heterocyclic derived M1 positive allosteric modulators

Scott D. Kuduk, Christina N. Di Marco, Victoria Cofre, Daniel R. Pitts, William J. Ray, Lei Ma, Marion Wittmann, Lone Veng, Matthew A. Seager, Kenneth Koeplinger, Charles D. Thompson, George D. Hartma

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 1.60 MB

english, 2010

20

Bradykinin B1 antagonists: SAR studies in the 2,3-diaminopyridine series

Scott D. Kuduk, Ronald K. Chang, Christina Ng, Kathy L. Murphy, Richard W. Ransom, Cuyue Tang, Thomayant Prueksaritanont, Roger M. Freidinger, Douglas J. Pettibone, Mark G. Bock

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 197 KB

english, 2005

21

5-Piperazinyl pyridine carboxamide bradykinin B1 antagonists

Scott D. Kuduk, Christina Ng Di Marco, Ronald K. Chang, Michael R. Wood, June J. Kim, Kathy M. Schirripa, Kathy L. Murphy, Richard W. Ransom, Cuyue Tang, Maricel Torrent, Sookhee Ha, Thomayant Prueksa

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2006

Langue:

english

Fichier:

PDF, 301 KB

english, 2006

22

α-Hydroxy amides as a novel class of bradykinin B1 selective antagonists

Michael R. Wood, Kathy M. Schirripa, June J. Kim, Scott D. Kuduk, Ronald K. Chang, Christina N. Di Marco, Robert M. DiPardo, Bang-Lin Wan, Kathy L. Murphy, Richard W. Ransom, Raymond S.L. Chang, Marie

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2008

Langue:

english

Fichier:

PDF, 135 KB

english, 2008

23

Bradykinin B1 receptor antagonists: An α-hydroxy amide with an improved metabolism profile

Scott D. Kuduk, Ronald K. Chang, Robert M. DiPardo, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone, Mark G. Bock

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2008

Langue:

english

Fichier:

PDF, 169 KB

english, 2008

24

Amiloride derived inhibitors of acid-sensing ion channel-3 (ASIC3)

Scott D. Kuduk, Christina N. Di Marco, Ronald K. Chang, Robert M. DiPardo, Sean P. Cook, Matthew J. Cato, Aneta Jovanovska, Mark O. Urban, Michael Leitl, Robert H. Spencer, Stefanie A. Kane, Mark T. B

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2009

Langue:

english

Fichier:

PDF, 3.04 MB

english, 2009

25

Amidine derived inhibitors of acid-sensing ion channel-3 (ASIC3)

Scott D. Kuduk, Ronald K. Chang, Jenny M.-C. Wai, Christina N. Di Marco, Victoria Cofre, Robert M. DiPardo, Sean P. Cook, Matthew J. Cato, Aneta Jovanovska, Mark O. Urban, Michael Leitl, Robert H. Spe

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2009

Langue:

english

Fichier:

PDF, 1021 KB

english, 2009

26

Corrigendum to “Pyridine containing M1 positive allosteric modulators with reduced plasma protein binding” [Bioorg. Med. Chem. Lett. 20 (2010) 657]

Scott D. Kuduk, Christina N. Di Marco, Victoria Cofre, Daniel R. Pitts, William J. Ray, Lei Ma, Marion Wittmann, Matthew A. Seager, Kenneth Koeplinger, Charles D. Thompson, George D. Hartman, Mark T.

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 102 KB

english, 2010

27

Hydroxy cycloalkyl fused pyridone carboxylic acid M1 positive allosteric modulators

Scott D. Kuduk, Robert M. DiPardo, Douglas C. Beshore, William J. Ray, Lei Ma, Marion Wittmann, Matthew A. Seager, Kenneth A. Koeplinger, Charles D. Thompson, George D. Hartman, Mark T. Bilodeau

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 808 KB

english, 2010

28

Heterocyclic fused pyridone carboxylic acid M1 positive allosteric modulators

Scott D. Kuduk, Christina N. Di Marco, Ronald K. Chang, William J. Ray, Lei Ma, Marion Wittmann, Matthew A. Seager, Kenneth A. Koeplinger, Charles D. Thompson, George D. Hartman, Mark T. Bilodeau

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 2.06 MB

english, 2010

29

Fused heterocyclic M1 positive allosteric modulators

Scott D. Kuduk, Christina N. Di Marco, Victoria Cofre, William J. Ray, Lei Ma, Marion Wittmann, Matthew A. Seager, Kenneth A. Koeplinger, Charles D. Thompson, George D. Hartman, Mark T. Bilodeau

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 834 KB

english, 2011

30

Quinolizidinone carboxylic acid selective M1 allosteric modulators: SAR in the piperidine series

Scott D. Kuduk, Ronald K. Chang, Christina N. Di Marco, William J. Ray, Lei Ma, Marion Wittmann, Matthew A. Seager, Kenneth A. Koeplinger, Charles D. Thompson, George D. Hartman, Mark T. Bilodeau

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 1.48 MB

english, 2011

31

Identification of non-amidine inhibitors of acid-sensing ion channel-3 (ASIC3)

Scott D. Kuduk, Ronald K. Chang, Christina N. Di Marco, Robert M. DiPardo, Sean P. Cook, Matthew J. Cato, Aneta Jovanovska, Mark O. Urban, Michael Leitl, Robert H. Spencer, Stefanie A. Kane, George D.

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 1.09 MB

english, 2011

32

Reversal of diastereoselection in the addition of Grignard reagents to chiral 2-pyridyl tert-butyl (Ellman) sulfinimines

Scott D. Kuduk, Robert M. DiPardo, Ronald K. Chang, Christina Ng, Mark G. Bock

Journal:

Tetrahedron Letters

Année:

2004

Langue:

english

Fichier:

PDF, 257 KB

english, 2004

33

Application of the thioimidate cyclopropane rearrangement to heterocyclic synthesis. Preparation of diaryl pyrrolines

Ronald K. Chang, Robert M. DiPardo, Scott D. Kuduk

Journal:

Tetrahedron Letters

Année:

2005

Langue:

english

Fichier:

PDF, 102 KB

english, 2005

34

Asymmetric addition reactions of Grignard reagents to chiral 2-trifluoromethyl tert-butyl (Ellman) sulfinimine–ethanol adducts

Scott D. Kuduk, Christina Ng Di Marco, Steven M. Pitzenberger, Nancy Tsou

Journal:

Tetrahedron Letters

Année:

2006

Langue:

english

Fichier:

PDF, 183 KB

english, 2006

35

Preparation of 4-heteroaryl-4-cyanopiperidines via SNAr substitution reactions

Ronald K. Chang, Christina N. Di Marco, Daniel R. Pitts, Thomas J. Greshock, Scott D. Kuduk

Journal:

Tetrahedron Letters

Année:

2009

Langue:

english

Fichier:

PDF, 2.03 MB

english, 2009

36

Preparation of 2,4,5-trisubstituted pyrazolo[4,3-c]quinolin-3-ones

Douglas C. Beshore, Robert M. DiPardo, Scott D. Kuduk

Journal:

Tetrahedron Letters

Année:

2010

Langue:

english

Fichier:

PDF, 931 KB

english, 2010

37

A highly efficient route to taxotere by the β-Lactam Synthon Method

Iwao Ojima, Chung Ming Sun, Martine Zucco, Young Hoon Park, Olivier Duclos, Scott Kuduk

Journal:

Tetrahedron Letters

Année:

1993

Langue:

english

Fichier:

PDF, 264 KB

english, 1993

38

Synthesis of 2,3-diaminodihydropyrroles via thioimidate cyclopropane rearrangement

Scott D Kuduk, Christina Ng, Ronald K Chang, Mark G Bock

Journal:

Tetrahedron Letters

Année:

2003

Langue:

english

Fichier:

PDF, 145 KB

english, 2003

39

Dianion equivalents corresponding to the polypropionate domain of epothilone B

Christina R. Harris, Scott D. Kuduk, Ken Savin, Aaron Balog, Samuel J. Danishefsky

Journal:

Tetrahedron Letters

Année:

1999

Langue:

english

Fichier:

PDF, 224 KB

english, 1999

40

Synthesis and evaluation of geldanamycin–testosterone hybrids

Scott D Kuduk, Christina R Harris, Fuzhong F Zheng, Laura Sepp-Lorenzino, Quathek Ouerfelli, Neal Rosen, Samuel J Danishefsky

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2000

Langue:

english

Fichier:

PDF, 160 KB

english, 2000

41

Synthesis and biological activity of 3′-alkyl- and 3′-alkenyl-3′-dephenyldocetaxels

Iwao Ojima, Olivier Duclos, Scott D. Kuduk, Chung-Ming Sun, John C. Slater, François Lavelle, Jean M. Veith, Ralph J. Bernacki

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1994

Langue:

english

Fichier:

PDF, 320 KB

english, 1994

42

N-acyl-3-hydroxy-β-lactams as key intermediates for taxotere and its analogs

Iwao Ojima, Martine Zucco, Olivier Duclos, Scott D. Kuduk, Chung Ming Sun, Young Hoon Park

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1993

Langue:

english

Fichier:

PDF, 282 KB

english, 1993

43

Synthesis and evaluation of geldanamycin-estradiol hybrids

Scott D. Kuduk, Fuzhong F. Zheng, Laura Sepp-Lorenzino, Neal Rosen, Samuel J. Danishefsky

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1999

Langue:

english

Fichier:

PDF, 339 KB

english, 1999

44

Structure–activity relationship study of taxoids for their ability to activate murine macrophages as well as inhibit the growth of macrophage-like cells

Iwao Ojima, Cecilia L Fumero-Oderda, Scott D Kuduk, Zhuping Ma, Fumiko Kirikae, Teruo Kirikae

Journal:

Bioorganic & Medicinal Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 662 KB

english, 2003

45

Diclofenac hydroxylation in monkeys: Efficiency, regioselectivity, and response to inhibitors

Cuyue Tang, Yulin Fang, Catherine Booth-Genthe, Yuhsin Kuo, Scott D. Kuduk, Tom H. Rushmore, Brian A. Carr

Journal:

Biochemical Pharmacology

Année:

2007

Langue:

english

Fichier:

PDF, 728 KB

english, 2007

46

Total Synthesis and Antitumor Activity of 12,13-Desoxyepothilone F: An Unexpected Solvolysis Problem at C15, Mediated by Remote Substitution at C21

Lee, Chul Bom, Chou, Ting-Chao, Zhang, Xiu-Guo, Wang, Zhi-Guang, Kuduk, Scott D., Chappell, Mark D., Stachel, Shawn J., Danishefsky, Samuel J.

Journal:

Journal of Organic Chemistry

Année:

2000

Langue:

english

Fichier:

PDF, 102 KB

english, 2000

47

Structural Requirements of Taxoids for Nitric Oxide and Tumor Necrosis Factor Production by Murine Macrophages

Teruo Kirikae, Iwao Ojima, Fumiko Kirikae, Zhuping Ma, Scott D. Kuduk, John C. Slater, Craig S. Takeuchi, Pierre-Yues Bounaud, Masayasu Nakano

Journal:

Biochemical and Biophysical Research Communications

Année:

1996

Langue:

english

Fichier:

PDF, 172 KB

english, 1996

48

2,3-Diaminopyridine Bradykinin B 1 Receptor Antagonists

Kuduk, Scott D., Ng, Christina, Feng, Dong-Mei, Wai, Jenny M.-C., Chang, Raymond S. L., Harrell, Charles M., Murphy, Kathy L., Ransom, Richard W., Reiss, Duane, Ivarsson, Magnus, Mason, Glenn, Boyce,

Journal:

Journal of Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 83 KB

english, 2004

49

Identification of Amides as Carboxylic Acid Surrogates for Quinolizidinone-Based M 1 Positive Allosteric Modulators

Kuduk, Scott D., Chang, Ronald K., Greshock, Thomas J., Ray, William J., Ma, Lei, Wittmann, Marion, Seager, Matthew A., Koeplinger, Kenneth A., Thompson, Charles D., Hartman, George D., Bilodeau, Mark

Journal:

ACS Medicinal Chemistry Letters

Année:

2012

Langue:

english

Fichier:

PDF, 369 KB

english, 2012

50

Synthetic and Immunological Studies on Clustered Modes of Mucin-Related Tn and TF O-Linked Antigens: The Preparation of a Glycopeptide-Based Vaccine for Clinical Trials against Prostate Cancer †

Kuduk, Scott D., Schwarz, Jacob B., Chen, Xiao-Tao, Glunz, Peter W., Sames, Dalibor, Ragupathi, Govindaswami, Livingston, Philip O., Danishefsky, Samuel J.

Journal:

Journal of the American Chemical Society

Année:

1998

Langue:

english

Fichier:

PDF, 577 KB

english, 1998